Development of a Highly Selective Plasmodium falciparum Proteasome Inhibitor with Anti-malaria Activity in Humanized Mice.

Wenhu Zhan, Hao Zhang, John Ginn, Annie Leung, Yi J Liu, Mayako Michino, Akinori Toita, Rei Okamoto, Tzu-Tshin Wong, Toshihiro Imaeda, Ryoma Hara, Takafumi Yukawa, Sevil Chelebieva, Patrick K. Tumwebaze, Maria Jose Lafuente-Monasterio, Maria Santos Martinez-Martinez, Jeremie Vendome, Thijs Beuming, Kenjiro Sato, Kazuyoshi AsoPhilip J. Rosenthal, Roland A. Cooper, Peter T Meinke, Carl F Nathan, Laura A Kirkman, Gang Lin

Research output: Contribution to journalArticlepeer-review

Original languageAmerican English
JournalDefault journal
Volume60
DOIs
StatePublished - Apr 19 2021

Keywords

  • Animals
  • Antimalarials
  • Drug Development
  • Malaria
  • Falciparum
  • Mice
  • Models
  • Molecular
  • Molecular Conformation
  • Parasitic Sensitivity Tests
  • Plasmodium falciparum
  • Proteasome Endopeptidase Complex
  • Proteasome Inhibitors

Disciplines

  • Life Sciences
  • Physical Sciences and Mathematics

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