Plasmodium falciparum Resistance to a Lead Benzoxaborole Due to Blocked Compound Activation and Altered Ubiquitination or Sumoylation.

Kirthana M. V. Sindhe, Wesley Wu, Jenny Legac, Yong-Kang Zhang, Eric E. Easom, Roland A. Cooper, Jacob J Plattner, Yvonne R. Freund, Joseph L. DeRisi, Philip J. Rosenthal

Research output: Contribution to journalArticlepeer-review

Original languageAmerican English
JournalDefault journal
Volume11
DOIs
StatePublished - Jan 28 2020

Keywords

  • malaria
  • Plasmodium falciparum
  • drug
  • benzoxaborole
  • resistance
  • PfPARE
  • ubiquitination
  • sumoylation
  • antimalarial agents
  • drug resistance evolution
  • drug resistance mechanisms

Disciplines

  • Medical Pharmacology
  • Medical Sciences

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